docetaxel anhydrous has been researched along with 6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one in 1 studies
Studies (docetaxel anhydrous) | Trials (docetaxel anhydrous) | Recent Studies (post-2010) (docetaxel anhydrous) | Studies (6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one) | Trials (6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one) | Recent Studies (post-2010) (6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one) |
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12,110 | 3,216 | 6,920 | 27 | 1 | 22 |
Protein | Taxonomy | docetaxel anhydrous (IC50) | 6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one (IC50) |
---|---|---|---|
Chain A, Tyrosine-protein kinase SYK | Homo sapiens (human) | 0.041 | |
Chain A, Tyrosine-protein kinase SYK | Homo sapiens (human) | 0.041 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Chain A, Tyrosine-protein kinase BTK | Homo sapiens (human) | 0.29 | |
Tyrosine-protein kinase JAK2 | Homo sapiens (human) | 0.006 | |
Tyrosine-protein kinase Lyn | Homo sapiens (human) | 0.732 | |
Proto-oncogene tyrosine-protein kinase receptor Ret | Homo sapiens (human) | 0.005 | |
Dipeptidyl peptidase 4 | Rattus norvegicus (Norway rat) | 0.041 | |
Tyrosine-protein kinase ZAP-70 | Homo sapiens (human) | 0.042 | |
Tyrosine-protein kinase SYK | Homo sapiens (human) | 0.167 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 1 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ | 1 |
1 other study(ies) available for docetaxel anhydrous and 6-[[5-fluoro-2-(3,4,5-trimethoxyanilino)-4-pyrimidinyl]amino]-2,2-dimethyl-4H-pyrido[3,2-b][1,4]oxazin-3-one
Article | Year |
---|---|
Identification of potent Yes1 kinase inhibitors using a library screening approach.
Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship | 2013 |